Work with Keykavous Parang | NotedSource
Professor
https://cv.notedsource.io/me/8OL4MD7R
Keykavous Parang
Professor
Research Expertise
Research in Drug Discovery
Drug Delivery
Nanotechnology
Organic Chemistry
Legacy Map
Full ViewPublications
Author index volume 10 (1990)
Statistics & Probability
Letters
1990
A Global Review on Short Peptides:
Frontiers and Perspectives
Molecules
2021
Self-assembly of peptides to
nanostructures
Org. Biomol. Chem.
2014
Nucleoside reverse transcriptase
inhibitors possess intrinsic
anti-inflammatory activity
Science
2014
Protein pyrophosphorylation by inositol
pyrophosphates is a posttranslational
event
Proceedings of the National Academy of
Sciences
2007
Cell‐Penetrating Homochiral Cyclic
Peptides as Nuclear‐Targeting Molecular
Transporters
Angewandte Chemie International
Edition
2011
Novel Approaches for Designing 5-O-Ester
Prodrugs of 3-Azido-2,3-dideoxythymidine
(AZT).
Current Medicinal Chemistry
2000
Impairment of TrkB-PSD-95 Signaling in
Angelman Syndrome
PLoS Biology
2013
Inhibitors of Protein Kinase Signaling
Pathways
Circulation
2004
Current Targets for Anticancer Drug
Discovery
Current Drug Targets
2003
Cyclic Cell-Penetrating Peptides as
Efficient Intracellular Drug Delivery
Tools
Molecular Pharmaceutics
2019
Designing bisubstrate analog inhibitors
for protein kinases
Pharmacology & Therapeutics
2002
Design and Biological Evaluation of
Cell-Penetrating Peptide–Doxorubicin
Conjugates as Prodrugs
Molecular Pharmaceutics
2013
Development of cytarabine prodrugs and
delivery systems for leukemia treatment
Expert Opinion on Drug Delivery
2010
Synthesis of
3-phenylpyrazolopyrimidine-1,2,3-triazole
conjugates and evaluation of their Src
kinase inhibitory and anticancer
activities
Bioorganic & Medicinal Chemistry
Letters
2011
A Review (Research and Patents) on
Jasmonic Acid and Its Derivatives
Archiv der Pharmazie
2014
Fatty acyl amide derivatives of
doxorubicin: Synthesis and in vitro
anticancer activities
European Journal of Medicinal
Chemistry
2011
Determination of the substrate-docking
site of protein tyrosine kinase C-terminal
Src kinase
Proceedings of the National Academy of
Sciences
2003
Antibacterial Activities of Amphiphilic
Cyclic Cell-Penetrating Peptides against
Multidrug-Resistant Pathogens
Molecular Pharmaceutics
2014
Synthesis, Anticancer Activities, and
Cellular Uptake Studies of Lipophilic
Derivatives of Doxorubicin Succinate
Journal of Medicinal Chemistry
2012
Enhanced Cellular Uptake of Short
Polyarginine Peptides through Fatty
Acylation and Cyclization
Molecular Pharmaceutics
2014
Cyclic Dipeptides: The Biological and
Structural Landscape with Special Focus on
the Anti-Cancer Proline-Based Scaffold
Biomolecules
2021
Cyclic Peptide-Capped Gold Nanoparticles
as Drug Delivery Systems
Molecular Pharmaceutics
2012
3-Substitued indoles: One-pot synthesis
and evaluation of anticancer and Src
kinase inhibitory activities
Bioorganic & Medicinal Chemistry
Letters
2011
Cyclic Peptide–Selenium Nanoparticles as
Drug Transporters
Molecular Pharmaceutics
2014
Thiazolyl N-benzyl-substituted acetamide
derivatives: Synthesis, Src kinase
inhibitory and anticancer activities
European Journal of Medicinal
Chemistry
2011
Protein Kinase Inhibitors in Drug
Discovery
Pharmaceutical Sciences
Encyclopedia
2010
Conformationally Constrained Peptide
Analogues of pTyr-Glu-Glu-Ile as
Inhibitors of the Src SH2 Domain Binding
Journal of Medicinal Chemistry
2004
Click chemistry inspired one-pot synthesis
of 1,4-disubstituted 1,2,3-triazoles and
their Src kinase inhibitory activity
Bioorganic & Medicinal Chemistry
Letters
2011
Synthesis and Antifungal Activities of
Myristic Acid Analogs
Archiv der Pharmazie
1996
Benzimidazoles as new scaffold of sirtuin
inhibitors: Green synthesis, in vitro
studies, molecular docking analysis and
evaluation of their anti-cancer properties
European Journal of Medicinal
Chemistry
2014
Copper catalyzed tandem oxidative C–H
amination/cyclizations: Direct access to
imidazo[1,2-a]pyridines
RSC Advances
2013
Carboxylic acid and phosphate ester
derivatives of fluconazole: synthesis and
antifungal activities
Bioorganic & Medicinal
Chemistry
2004
Efficient Delivery of Cell Impermeable
Phosphopeptides by a Cyclic Peptide
Amphiphile Containing Tryptophan and
Arginine
Molecular Pharmaceutics
2013
Copper triflate-mediated synthesis of
1,3,5-triarylpyrazoles in [bmim][PF6]
ionic liquid and evaluation of their
anticancer activities
RSC Advances
2013
Synthesis and evaluation of novel
benzimidazole derivatives as sirtuin
inhibitors with antitumor activities
Bioorganic & Medicinal
Chemistry
2014
A Simple and Efficient Synthesis of
2,3-Diarylnaphthofurans Using Sequential
Hydroarylation/Heck Oxyarylation
Organic Letters
2013
In vitro antiviral activities of myristic
acid analogs against human
immunodeficiency and hepatitis B viruses
Antiviral Research
1997
Inhibition of N-Methyl-d-aspartate-induced
Retinal Neuronal Death by Polyarginine
Peptides Is Linked to the Attenuation of
Stress-induced Hyperpolarization of the
Inner Mitochondrial Membrane Potential
Journal of Biological Chemistry
2015
Synthesis of novel ciprofloxacin analogues
and evaluation of their anti-proliferative
effect on human cancer cell lines
Bioorganic & Medicinal Chemistry
Letters
2013
Synthesis and Biological Evaluation of
Fatty Acyl Ester Derivatives of
(−)-2′,3′-Dideoxy-3′-thiacytidine
Journal of Medicinal Chemistry
2012
Emtricitabine Prodrugs with Improved
Anti-HIV Activity and Cellular Uptake
Molecular Pharmaceutics
2012
Self-assembled surfactant cyclic peptide
nanostructures as stabilizing agents
Soft Matter
2013
Synthesis and evaluation of fatty acyl
ester derivatives of cytarabine as
anti-leukemia agents
European Journal of Medicinal
Chemistry
2010
Development of photo‐crosslinking reagents
for protein kinase–substrate interactions
FEBS Letters
2002
Cytoplasmic synthesis of endogenous
Alu
complementary DNA via reverse
transcription and implications in
age-related macular degeneration
Proceedings of the National Academy of
Sciences
2021
Synthesis and antiproliferative activities
of doxorubicin thiol conjugates and
doxorubicin-SS-cyclic peptide
European Journal of Medicinal
Chemistry
2019
Facile, Regio- and Diastereoselective
Synthesis of Spiro-Pyrrolidine and
Pyrrolizine Derivatives and Evaluation of
Their Antiproliferative Activities
Molecules
2014
4-Aryl-4H-naphthopyrans derivatives:
one-pot synthesis, evaluation of Src
kinase inhibitory and anti-proliferative
activities
DARU Journal of Pharmaceutical
Sciences
2012
Probing the Catalytic Mechanism of the
Insulin Receptor Kinase with a
Tetrafluorotyrosine-containing Peptide
Substrate
Journal of Biological Chemistry
2000
Ionic Liquid as Soluble Support for
Synthesis of 1,2,3-Thiadiazoles and
1,2,3-Selenadiazoles
The Journal of Organic Chemistry
2012
Synthesis, Analysis, in Vitro
Characterization, and in Vivo Disposition
of a Lamivudine–Dextran Conjugate for
Selective Antiviral Delivery to the Liver
Bioconjugate Chemistry
2007
Comparative Antiviral Activity of
Remdesivir and Anti-HIV Nucleoside Analogs
against Human Coronavirus 229E (HCoV-229E)
Molecules
2020
Synthesis of
4-aryl-6-indolylpyridine-3-carbonitriles
and evaluation of their antiproliferative
activity
Tetrahedron Letters
2014
Cyclic Peptide-Capped Gold Nanoparticles
for Enhanced siRNA Delivery
Molecules
2014
Selective Diphosphorylation,
Dithiodiphosphorylation,
Triphosphorylation, and
Trithiotriphosphorylation of Unprotected
Carbohydrates and Nucleosides
Organic Letters
2005
Reactions of Solid-Supported Reagents and
Solid Supports with Alcohols and Phenols
through Their Hydroxyl Functional Group
Journal of Combinatorial
Chemistry
2003
Docking-based Substrate Recognition by the
Catalytic Domain of a Protein Tyrosine
Kinase, C-terminal Src Kinase (Csk)
Journal of Biological Chemistry
2006
Synthesis and Antiproliferative Activities
of Conjugates of Paclitaxel and
Camptothecin with a Cyclic
Cell-Penetrating Peptide
Molecules
2019
Design, Synthesis, and Evaluation of
Amphiphilic Cyclic and Linear Peptides
Composed of Hydrophobic and
Positively-Charged Amino Acids as
Antibacterial Agents
Molecules
2018
Synthesis and Evaluation of Antimicrobial
Activity of [R4W4K]-Levofloxacin and
[R4W4K]-Levofloxacin-Q Conjugates
Molecules
2017
Synthesis and Evaluation of Tripodal
Peptide Analogues for Cellular Delivery of
Phosphopeptides
Journal of Medicinal Chemistry
2007
4-Aryl-4H-Chromene-3-Carbonitrile
Derivatives: Evaluation of Src Kinase
Inhibitory and Anticancer Activities
Medicinal Chemistry
2011
Surface Decorated Gold Nanoparticles by
Linear and Cyclic Peptides as Molecular
Transporters
Molecular Pharmaceutics
2013
ChemInform Abstract: 3‐Substituted
Indoles: One‐Pot Synthesis and Evaluation
of Anticancer and Src Kinase Inhibitory
Activities.
ChemInform
2011
Solid-Phase Synthesis of Symmetrical
5‘,5‘-Dinucleoside Mono-, Di-, Tri-, and
Tetraphosphodiesters
Organic Letters
2007
Hydrophobicity drives the cellular uptake
of short cationic peptide ligands
European Biophysics Journal
2011
Synthesis and Structure−Activity
Relationships of Linear and
Conformationally Constrained Peptide
Analogues of CIYKYY as Src Tyrosine Kinase
Inhibitors
Journal of Medicinal Chemistry
2006
A Solid Phase Reagent for the Capture
Phosphorylation of Carbohydrates and
Nucleosides
Organic Letters
2001
Cationic Cell-Penetrating Peptides Are
Potent Furin Inhibitors
PLOS ONE
2015
Amphiphilic Bicyclic Peptides as Cellular
Delivery Agents
ChemMedChem
2014
Synthesis and biological evaluation of
fatty acyl ester derivatives of
2′,3′-didehydro-2′,3′-dideoxythymidine
Bioorganic & Medicinal Chemistry
Letters
2011
Src kinase inhibitors: an emerging
therapeutic treatment option for prostate
cancer
Expert Opinion on Investigational
Drugs
2010
Membrane-Active Cyclic Amphiphilic
Peptides: Broad-Spectrum Antibacterial
Activity Alone and in Combination with
Antibiotics
Journal of Medicinal Chemistry
2022
Nano drug delivery systems as promising
tools for cancer therapy
Journal of NanoScience Technology
2022
Probing the Communication between the
Regulatory and Catalytic Domains of a
Protein Tyrosine Kinase, Csk
Biochemistry
2005
Synthesis and Evaluation of
3‐Phenylpyrazolo[3,4‐d]pyrimidine‐Peptide
Conjugates as Src Kinase Inhibitors
ChemMedChem
2007
Conformational Basis for SH2-Tyr(P)527
Binding in Src Inactivation
Journal of Biological Chemistry
2006
Bisubstrate analog probes for the insulin
receptor protein tyrosine kinase:
Molecular yardsticks for analyzing
catalytic mechanism and inhibitor design
Bioorganic Chemistry
2005
ATP-phosphopeptide conjugates as
inhibitors of Src tyrosine kinases
Bioorganic & Medicinal
Chemistry
2004
Novel pH-Sensitive Cyclic Peptides
Scientific Reports
2016
Cysteine and arginine-rich peptides as
molecular carriers
Bioorganic & Medicinal Chemistry
Letters
2016
Base-Mediated Chemo- and Stereoselective
Addition of 5-Aminoindole/Tryptamine and
Histamines onto Alkynes
The Journal of Organic Chemistry
2013
2,6‐hexadecadiynoic acid and
2,6‐nonadecadiynoic acid: Novel
synthesized acetylenic fatty acids as
potent antifungal agents
Lipids
2006
Structural Basis for Domain–Domain
Communication in a Protein Tyrosine
Kinase, the C-terminal Src Kinase
Journal of Molecular Biology
2006
Recent advances in the discovery of Src
kinase inhibitors
Expert Opinion on Therapeutic
Patents
2005
Design of tetrapeptide ligands as
inhibitors of the Src SH2 domain
Bioorganic & Medicinal
Chemistry
2004
Antibiotics-Peptide Conjugates Against
Multidrug-resistant Bacterial Pathogens
Current Topics in Medicinal
Chemistry
2019
Design, synthesis, and evaluation of
chitosan conjugated GGRGDSK peptides as a
cancer cell-targeting molecular
transporter
International Journal of Biological
Macromolecules
2016
Synthesis and Anti-HIV Activities of
Glutamate and Peptide Conjugates of
Nucleoside Reverse Transcriptase
Inhibitors
Journal of Medicinal Chemistry
2012
Cyclic Peptide Containing Hydrophobic and
Positively Charged Residues as a Drug
Delivery System for Curcumin
Current Drug Delivery
2016
On water: catalyst-free chemoselective
synthesis of highly functionalized
tetrahydroquinazolines from
2-aminophenylacrylate
Green Chemistry
2015
Solid-Phase Reagents for Selective
Monophosphorylation of Carbohydrates and
Nucleosides
The Journal of Organic Chemistry
2005
TrkB-enhancer facilitates functional
recovery after traumatic brain injury
Scientific Reports
2017
Synthesis and in Vitro Characterization of
Novel Dextran–Methylprednisolone
Conjugates with Peptide Linkers: Effects
of Linker Length on Hydrolytic and
Enzymatic Release of Methylprednisolone
and its Peptidyl Intermediates
Journal of Pharmaceutical
Sciences
2008
Synthesis and evaluation of c-Src kinase
inhibitory activity of pyridin-2(1H)-one
derivatives
Bioorganic Chemistry
2014
Ionic Liquid-Supported Synthesis of
Sulfonamides and Carboxamides
ACS Combinatorial Science
2011
Bilayer disruption and liposome
restructuring by a homologous series of
small Arg-rich synthetic peptides
Colloids and Surfaces B:
Biointerfaces
2010
Amphiphilic Peptides for Efficient siRNA
Delivery
Polymers
2019
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